/hrt/feminizing/estradiol-oral
Estradiol (Oral)
[estradiol]Rev: 2025.12
Summary
An oral form of Estradiol, commonly used by those with a fear of needles.
DESCRIPTION
Oral estradiol is a bioidentical form of the primary female sex hormone estrogen, typically administered as estradiol hemihydrate or estradiol valerate tablets.
DOSING GUIDELINES
| Route | Dose Range | Frequency | Target Levels |
|---|---|---|---|
| Oral / Sublingual/Buccal | 2mg – 8mg | Daily | 100-300pg/mL |
DETAILED NOTES
Oral / Sublingual/Buccal
2mg-6mg must be taken with an anti-androgen, monotherapy levels (8mg daily) do not need an anti-androgen to suppress testosterone.
WHERE TO BUY
LIVE STOCKSublingual Estradiol Oil Dropper 30mL 20mg/mL20mg/mL
Open Gate LabsCOMMUNITY TRUSTED• oil dropper• 30mL
$80.00IN STOCK
Estrabet (Estradiol Hemihydrate) 2mg - 28 Tablets2mg
DashPCTUNVERIFIED• Tablet• 28 tablets
$12.00IN STOCK
Estradiol Valerate (EV, Ediol V) 132 - 10mg/ml 20ml10mg/ml
Dragon OrdnanceUNVERIFIED• Injectable• 20ml
$23.00IN STOCK
Estraheal 2mg - 28 Tablets (Estradiol)2mg
AipctshopUNVERIFIED• Tablet• 28 tablets
$5.00IN STOCK
Estrana tapes 0.72 mg0.72mg
Japan Health Center (Bio-Japan)UNVERIFIED• Patch• 70 sheets
$189IN STOCK
Estrofem 2 mg2mg
FavskinhouseUNVERIFIED• Tablet• 28 tablets
$20IN STOCK
Estrofem 2mg2mg
Inhouse PharmacyUNVERIFIED• Tablet• 28 tablets
$42IN STOCK
Progydol 2mg - 28 Tablet (Estradiol Valerate)2mg
AipctshopUNVERIFIED• Tablet• 28 tablets
$6.25IN STOCK
Progynova (Estradiol Valerate) - 2mg (28 Tablets)2mg
4NRX PharmacyUNVERIFIED• Tablet• 28 tablets
£16.10IN STOCK
Progynova 2 mg2mg
FavskinhouseUNVERIFIED• Tablet• 28 tablets
$12.90IN STOCK
Progynova 2mg2mg
Inhouse PharmacyUNVERIFIED• Tablet• 84 tablets
$52IN STOCK
Progynova 2mg (Estradiol Valerate) - 28 Tablets2mg
All Day ChemistUNVERIFIED• Tablet• 28 tablets
$11.00IN STOCK
Progynova (Estradiol Valerate) - 1mg (28 Tablets)1mg
4NRX PharmacyUNVERIFIED• Tablet• 28 tablets
£8.92PRE-ORDER
l'estrogel 0.06%0.06%
Japan Health Center (Bio-Japan)UNVERIFIED• Gel• 80g
$79OUT OF STOCK
Estradiol oral2mg/4mg
Otokonoko PharmaceuticalsCAUTION• tablet• 100 pills
$50.00 – $95.00OUT OF STOCK
Stock and prices updated automatically. Click to visit supplier.
Rev: 2025.12hrt.fm